| Patents for C07D 451 - Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.02,4] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof (5,273) |
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| 08/09/2007 | WO2007088514A1 Secondary amines as renin inhibitors |
| 08/09/2007 | WO2007054784A8 An improved process for the preparation of granisetron hydrochloride |
| 08/09/2007 | US20070185156 3-exo-(5-chlorobiphenyl-3-yloxy)-8-azabicyclo[3.2.1]octane; exo 5-(8-azabicyclo[3.2.1]oct-3-yloxy)biphenyl-3-carbonitrile; depression, pain |
| 08/09/2007 | US20070185155 1-(2-{[(3-fluorophenyl)methyl]oxy}ethyl)-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octane bromide; muscle relaxants, respiratory system disorders; asthma, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis |
| 08/09/2007 | US20070185148 M3 muscarinic acetylchoine receptor antagonists |
| 08/09/2007 | CA2637546A1 Secondary amines as renin inhibitors |
| 08/09/2007 | CA2635814A1 Amido compounds and their use as pharmaceuticals |
| 08/08/2007 | EP1487832B1 Micronized crystalline tiotropium bromide |
| 08/07/2007 | CA2302943C Phthalazine compounds and therapeutic agents for erectile dysfunction |
| 08/02/2007 | WO2007086554A1 Tropane compound and pharmaceutical composition containing the same as active ingredient |
| 08/02/2007 | US20070179158 2,6-Disubstituted piperiddines as modulators |
| 08/01/2007 | EP1487822B1 Pyrrole-2,5-dione derivatives and their use as gsk-3 inhibitors |
| 08/01/2007 | EP1484327B1 Nitrogenous heterocyclic compound and medicine thereof |
| 08/01/2007 | CN101010320A Aminotropane derivatives, preparation thereof and therapeutic use thereof |
| 08/01/2007 | CN101010309A Oxopiperidine derivatives, preparation and therapeutic use thereof |
| 07/31/2007 | US7250426 acid addition salt of optionally substituted 5-[2-(indan-2-ylamino-1-hydroxyethyl)]-8-hydroxyquinolone; treating respiratory disorders, especially asthma and COPD |
| 07/31/2007 | US7250425 Substituted in the 2 position with phenoxy(or thio)methyl- or naphthyloxy(or thio)methyl- and in the 3 position with alkyl, phenyl-, or naphthyl-, e.g., 2R,3S)-2-(2,3-Dichlorophenoxymethyl)-8-methyl-3-(3-chlorophenyl)-8-aza-bicyclo[3.2.1]octane |
| 07/26/2007 | WO2007058971A3 Soft anticholinergic esters |
| 07/26/2007 | US20070173646 e.g. 4-[cyano(di-2-thienyl)methyl]-1-[3-(phenyloxy)propyl]-1-azoniabicyclo[2.2.2]octane bromide; muscle relaxants, respiratory system disorders; asthma, emphysema, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis |
| 07/25/2007 | EP1809626A2 Aryl substituted 8-azabicyclo[3.2.1]octane compounds as ligands of the melanin concentrating hormone receptor |
| 07/25/2007 | EP1355873B1 Pleuromutilin derivatives with antimicrobial activity |
| 07/25/2007 | CN101006057A Novel piperidine/8-azabicyclo [3.2.1] octan derivatives as moduilators of chemokine receptor CCR5 |
| 07/25/2007 | CN101005842A Modulators of muscarinic receptors |
| 07/24/2007 | US7247643 8-aza-bicyclo (3.2.1) octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 07/24/2007 | US7247629 Antitumoral analogs of et-743 |
| 07/19/2007 | WO2007081995A2 Urotensin ii receptor antagonists |
| 07/19/2007 | WO2007081890A2 Production of dolasetron |
| 07/19/2007 | WO2007081889A2 Production of dolasetron |
| 07/19/2007 | US20070167627 Benzoquinolizine-2-carboxylic acid arginine salt tetrahydrate |
| 07/18/2007 | EP1808435A1 Technical synthesis method for producing tropenol |
| 07/18/2007 | EP1807423A2 Quinolinone-carboxamide compounds |
| 07/18/2007 | EP1807422A1 5-ht4 receptor agonist compounds |
| 07/18/2007 | CN101001855A Novel method for producing tiotropium salts |
| 07/18/2007 | CN100999521A Crystal anti-choline medicine thiatropic bromoammonium |
| 07/17/2007 | US7244742 Pharmaceutical compositions for inhalation containing an anticholinergic, corticosteroid and betamimetic |
| 07/12/2007 | WO2007079239A2 Bicyclic nitrogen compounds as modulators of ghrelin receptor and uses thereof |
| 07/12/2007 | WO2007079078A1 Diamine derivatives as inhibitors of leukotriene a4 hydrolase |
| 07/12/2007 | WO2007078251A1 Compounds |
| 07/12/2007 | WO2007077949A1 Heterocyclic janus kinase 3 inhibitors |
| 07/12/2007 | WO2007024651A3 Bridged n-bicyclic sulfonamido inhibitors of gamma secretase |
| 07/12/2007 | US20070161641 2-(4-thieno[2,3-d]isoxazol-3-yl-piperidin-1-ylmethyl)-(2R,3R)-cyclopropanecarboxylic acid (trans4-methyl-cyclohexyl)-amide; psychological disorders, neurodegenerative diseases, antidepressant; drug abuse, sleep disorders |
| 07/12/2007 | DE60125335T2 Azacyclische verbindungen zur verwendung in der behandlung von mit serotonin verwandten krankheiten Azacyclic compounds for use in the treatment of serotonin-related diseases |
| 07/12/2007 | CA2635850A1 Heterocyclic janus kinase 3 inhibitors |
| 07/10/2007 | US7241745 Pyridyl alkene and pyridyl alkine acid amides as cytostatics and immunosupressives |
| 07/05/2007 | WO2007075858A2 Novel forms of tiotropium bromide and processes for preparation thereof |
| 07/05/2007 | WO2007075838A2 Pure and stable tiotropium bromide |
| 07/05/2007 | WO2007016639A3 M3 muscarinic acetylcholine receptor antagonists |
| 07/05/2007 | US20070155781 ipratropium/flutropium/tiotropium derivatives; anticholinergic agent; linked at NO or NO2 group, or group which stimulates endogenous production of NO; beneficial therapeutic effects; asthma, respiratory disorder, cystic fibrosis; synergistic with NO release agent or substrate for nitric oxide synthase |
| 07/05/2007 | US20070155780 Stabilized composition containing 4-amino-5-chloro-n-[(1r, 3r, 5s)-8-methyl-8-azabicyclo[3.2.1]oct-3-y1]-2-[1-methylbut-2-ynyloxy]benzamide |
| 07/05/2007 | US20070155721 inflammatory conditions, allergies, autoimmune diseases, chronic pain, graft rejection, cancers which involve leukocyte filtration, stenosis or restenosis, atherosclerosis, rheumatoid arthritis, osteoarthritis; e.g. 4-Isobutoxy-1H-indole-2-carboxylic acid [4-(2-azepan-1-yl-ethyl)-phenyl]-amide |
| 07/05/2007 | CA2627729A1 Novel forms of tiotropium bromide and processes for preparation thereof |
| 07/05/2007 | CA2620142A1 Pure and stable tiotropium bromide |
| 07/04/2007 | EP1644343B1 5-substituted quinazolinone derivatives |
| 07/04/2007 | EP1375496B1 N-aryl-substituted cyclic amine derivative and medicine containing the same as active ingredient |
| 07/04/2007 | CN1990486A N-glycyl-pyrrolidine-2-nitrile and its use as DDP-IV enzyme inhibitor |
| 07/04/2007 | CN1990469A Pyrrolidines as dipeptidyl peptidase inhibitors |
| 07/04/2007 | CN1990468A Pyrrolidines as dipeptidyl peptidase inhibitors |
| 07/04/2007 | CN1324025C Tropane derivatives as CCR5 modulators |
| 07/03/2007 | US7238720 Pharmaceutical use of N-carbamoylazole derivatives |
| 07/03/2007 | US7238688 For therapy of allergy, allergy-induced airway responses, congestion, hypotension, cardiovascular disease, hypotension, diseases of the GI tract, hyper and hypo motility and acidic secretion of the gastrointestinal tract, obesity, sleep |
| 06/28/2007 | WO2007071400A1 Pyrazine derivatives as epithelial sodium channel blocker |
| 06/28/2007 | US20070149562 Oxopiperidine derivatives, preparation and therapeutic use thereof |
| 06/28/2007 | CA2630889A1 Pyrazine derivatives as epithelial sodium channel blocker |
| 06/21/2007 | US20070142377 Pyridyl Alkene and Pyridyl Alkine-Acid Amides as Cytostatics and Immunosuppressives |
| 06/21/2007 | US20070142351 Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands |
| 06/21/2007 | DE102005059602A1 Verfahren zur Mikronisierung Process for the micronization |
| 06/20/2007 | EP1797088A1 Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 06/20/2007 | CN1982309A Industrial synthesis method for producing tropenol |
| 06/14/2007 | US20070135505 Aralkyl ester soft drugs |
| 06/14/2007 | US20070135478 3-(2-Benzyl-2-hydroxy-3-phenyl-propylidene)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane iodide; muscle relaxants, respiratory system disorders; asthma, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis |
| 06/14/2007 | US20070135423 E-fluoro-4-(pyridin-2-yl)-piperidine-1-carboxamide derivatives and related compounds which modulate the function of the vanilloid-1 receptor (vr1) for the treatment of pain |
| 06/13/2007 | EP1794164A2 Bridged piperazine and piperidine derivatives as ccr1 antagonists |
| 06/13/2007 | EP1794158A2 Method for producing tiotropium salts and silicon derivatives as intermediates |
| 06/12/2007 | US7230001 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof |
| 06/12/2007 | CA2249410C Sigma-2 receptors as biomarkers of tumor cell proliferation |
| 06/07/2007 | US20070129397 Ester derivatives |
| 06/07/2007 | US20070129396 Muscarinic acetylcholine receptor antagonists |
| 06/06/2007 | EP1791838A2 Process for preparing substituted 8-azabicyclo[3.2.1] octan-3-ols |
| 06/06/2007 | CN1976911A Arylphenylamino-, arylphenylamide-, and arylphenylether-sulfide derivatives |
| 05/31/2007 | WO2007037518A9 Mutilin derivative and pharmaceutical composition containing the same |
| 05/31/2007 | WO2007030089A8 Tricyclic delta- opioid modulators |
| 05/31/2007 | CA2630222A1 Carbamate compounds as 5-ht4 receptor agonists |
| 05/30/2007 | EP1789404A2 Substituted n-arylsulfonylheterocyclic amines as gamma-secretase inhibitors |
| 05/29/2007 | US7223776 Compounds with anti-bacterial activity |
| 05/24/2007 | WO2007059021A1 Soft anticholinergic zwitterions |
| 05/24/2007 | WO2006021655A8 Oxopiperidine derivatives, preparation and therapeutic use thereof |
| 05/24/2007 | CA2627982A1 Soft anticholinergic esters |
| 05/23/2007 | EP1787992A1 Pyrrolopyrimidine and pyrrolopyridine derivatives substituted with cyclic amino group |
| 05/23/2007 | EP1787984A2 Azacyclic compounds for use in the treatment of serotonin related diseases |
| 05/23/2007 | EP1786809A2 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
| 05/23/2007 | EP0859777B1 8-azabicyclo(3.2.1)oct-2-ene derivatives, their preparation and use |
| 05/22/2007 | CA2157579C Heterocyclic compounds, their use and preparation |
| 05/18/2007 | WO2007054784A1 An improved process for the preparation of granisetron hydrochloride |
| 05/18/2007 | WO2007054531A1 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 05/18/2007 | CA2629237A1 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 05/16/2007 | EP1785422A1 Micronised crystalline tiotropium bromide |
| 05/16/2007 | EP1785421A1 Tropan compound |
| 05/16/2007 | EP1434485B1 Nicotinic acid-heterocyclyl-amides and analogous pyrimidine derivatives for use as pesticides |
| 05/16/2007 | CN1962657A 2-beta- carbomethoxy-3 beta-(4- chlorphenyl) tropane synthesis method |
| 05/15/2007 | US7217716 Such as 4-((methyl-pyrimidin-2-ylamino)-methyl)-piperidine-1-carboxylic acid benzyl ester; useful for pain relief; treating migraine, depression, anxiety, schizophrenia, Parkinson's disease, and stroke; N-methyl-D-aspartate NR2B antagonists |